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| 发布时间：2019-05-20 访问次数:888 作者: |
 contact information
office: room 1035b, researching building 18 email: jyf@ecust.edu.cn office phone: 86 21 6425 3314 office fax: 86 21 6425 3314
education 2001.06 ph.d. applied chemistry, china university of mining technology, beijing, p. r. china 1992.06 m.eng. fine chemical engineering, east china university ofscience&technology, shanghai, p. r. china 1984.06 b.s. chemical education, , wuhu, p. r. china
professional experience 2007.9-now professor, department of pharmaceutical engineering, school of pharmacy, ecust 2009.03-2010.03 visiting scholar, department of chemistry and chemical biology, university of new mexico 2003.12-2007.8 associate professor, department of pharmaceutical engineering, ecust 2001.12-2003.11 postdoc fellow, institute of materia medica, peking union medical college, chinese academy of medical sciences 1996.11-2001.10 associate professor, school of chemical engineering, china university of mining technology, xuzhou, p. r. china 1992.8-1996.10 a r , anhui institute of materia medica, hefei, p. r. china
research interests organic chemistry - developing new synthetic methods, practical catalysts and efficient strategies for the synthesis of valuable fine chemicals and pharmaceuticals. green chemistry - designing new synthetic pathways for sustainable synthesis and production.
publication hu yh, shao ly, ji yf.* palladium-catalyzed arylation of aromatic amides directed by 2-amino-5-cholophenyl-1h-pyrazole auxiliary. synlett 2018-6-15, accepted. shao ly, xing lh,guo y, yu kk, wang w, liu hw, liao dh, ji yf.* catalytic cascade access to biaryl-2-methyl acetates from pyruvate o-arylmethyl ketoximes via the palladium-catalyzed c(sp2)–h bond arylation and c–o bond solvolysis. adv. synth. catal. 2018, doi 10.1002/adsc.201800216, published online. qiao wl, shao ly, hu yh, xing lh, deng kz, liao dh, dao-hua liao, ji yf.* palladium-catalyzed csp3–h bond mono-aroyloxylation of o-alkyl substituted 2,4,6-tri- methoxybenzaldoxime ethers. synlett2018, 29, 1249–1255. guo y, shao ly, yu kk, hu yh, liu hw,* liao dh, ji yf*. palladium-catalyzed site-selective direct olefination of 6-electron-withdrawing group substitued 3-arylbenzo[d]isoxazoles. org. chem. front.2017, 4, 1962–1966. guo y, yu kk, xing lh, liu hw, wang w,* ji yf*. palladium-catalyzed divergent regioselective homocoupling and hydroxylation of 3-arylbenzo[d]isoxazoles. adv. synth. catal. 2017, 359(3), 410–418. shao ly, li c,guo y, yu kk,zhao fy,qiao wl, liu hw, liao dh,* ji yf*. pd-catalyzed direct oxidative mono-aroyloxylation of o-aralkyl substituted acetoxime ethers. rsc advances, 2016, 6, 78875–78880. yu, kk, guo y, hu yh, xu z, liu hw, liao dh,* ji yf*. pd-catalyzed diverse mono-acyloxylation of 5-alkyl-4-aryl-thiazole-2-carboxylates. asian j. org. chem. 2016, 5, 1219–1224. ding j, guo y, shao ly, zhao fy, liao dh, liu hw*, ji yf*. palladium-catalyzed multi-acetoxylation of 1,3-disubstituted 1h-pyrazole-5-carboxylates via direct c(sp2)−h or c(sp3)−h bond activation. chin. chem. lett.2016, 27, 1617–1621. fan xm,guo y, li yd,yu kk, liu hw, liao dh, ji yf*.pd-catalyzed late-stage mono-acetoxylation and mono-iodination of 4-alkyl-1,5-diaryl-1h-pyrazole-3-carboxylates via direct csp2-h bond activation. asian j. org. chem. 2016, 5, 499–505. zhang zn, huang jg, zhai jj, guo y, ji yf*. copper(ii)-catalyzed oxidative esterification of substituted p-cresols under ligand- and additive-free conditions. synlett2015, 26, 2145–2150. guo y, li yd, chen c, zhao jh, liu hw, liao dh, ji yf*. a practical ligand-free copper(i) bromide-catalyzed fluoroalkoxylation of unactivated aryl bromides. res. chem. intermediat. 2016, 42, 2525–2537. huang jg, guo y, li yd, liu hw,* liao dh, ji yf*. undecorated cu(oac)2-catalyzed c(sp3)–c(sp3) bond formation through a para-hydroxyl group-triggered remote benzylic c(sp3)–h bond functionalization. eur. j. org. chem.2015, 5334–5338. guo y, fan xm, nie m, liu hw, liao dh, pan xd,* ji yf*. practical ligand-free cu-catalyzed short-chain alkoxylation of unactivated aryl bromides. eur. j. org. chem.2015, 4744–4755. guo y, chen c, liu hw,* zhao jh, zheng, yl, ji yf*. a ligand-free, powerful and practical method for methoxylation of unactivated aryl bromides by use of cucl/hcoome/meona/meoh system. res. chem. intermediat.2015, 41, 8651–8664. zhai jj, gu ch, guo y, liao dh, zhu dr, ji yf*. one-pot synthesis of highly substituted 1h-pyrazole-5-carboxylates from 4-aryl-2,4-diketoesters and arylhydrazines. j. heterocyclic chem.2016, 53, 840–848. huang jg, guo y, jiang ja, liu hw, ji yf*. an eco-friendly co(oac)2-catalyzed aerobic oxidation of 4-benzylphenols into 4-hydroxybenzophenones. res. chem. intermediat.2015, 41, 7115–7124. jiang ja, chen c, guo y, liao dh, pan xd, ji yf*. a highly efficient approach to vanillin starting from 4-cresol. green chem.2014, 16, 2807–2814. guch, zhai jj, jiang ja, liu hw, wang l, zhu dr, ji yf*. an efficient one-pot synthesis of aryl-substituted 1-(thiazol-2-yl)-1h-pyrazole-3-carboxylates via a hantzsch synthesis-knorr reaction sequence. chin. j. chem.2014, 32, 179–190. jiang ja, chen c, huang jg, liu hw, cao s, ji yf*. cu(oac)2-catalyzedremote benzylic c(sp3)–hoxyfunctionalization for c=o formation directed by the hindered para-hydroxyl group with ambient air as terminal oxidant under ligand- and additive-free conditions. green chem.2014, 16, 1248–1254. jiang ja, du jl, liao dh, wang zg, ji yf*. efficient co(oac)2-catalyzed aerobic oxidation of ewg-substituted 4-cresols to access 4-hydroxybenzaldehydes. tetrahedron lett. 2014, 55, 1406– 1411. jiang ja, du jl, zhang zn, zhai jj, ji yf*. an environmentally friendly and highly efficient co(oac)2-catalyzed aerobic oxidation to access 2,6-di-electron-donating group substituted 4-hydroxybenzaldehydes. syn. commun. 2014, 44, 1430–1440. zhai jj, gu ch, jiang ja, zhang sl, liao dh, wang l,zhu dr, ji yf*. a one- pot approach to ethyl 1,4,5-triaryl-1h-pyrazole-3-carboxylates via an improved claisen condensation-knorr reaction sequence. chin. j. chem.2013, 31, 1526–1538. zhai jj, jiang ja, zhang sl, chen c, liu hw, liao dw, ji yf*. stereoselective or exclusive synthesis of ethyl z-2-(2-substituted-thiazol-4-yl)pent-2-enoates from ethyl e/z-2-(2-bromoacetyl) pent-2-enoate. synlett 2013, 24, 1399–1404. huang wb, guo y, jiang ja, pan xd, liao dh, ji yf*. an efficient strategy for protecting dihydroxyl groups of catechols. synlett 2013, 24, 741–746. jiang ja, huang wb, zhai jj, liu hw, cai q, xu lx, wang w, ji yf*. “one-pot” synthesis of 4-substituted 1,5-diaryl-1h-pyrazole-3-carboxylates via lithium tert-butoxide-mediated sterically hindered claisen condensation and knorr reaction. tetrahedron 2013, 69, 627–635. jiang ja, ji yf*. alternative synthesis of apixaban (bms-562247), an inhibitor of blood coagulation factor xa. syn. commun. 2013, 43, 72–79. huang wb, du cy, jiang ja, ji yf*. concurrent synthesis of vanillin and isovanillin. res. chem. intermediat.2013, 39(6), 2849–2856. ji yf*, jiang ja, liu hw, liao dh, wei xy. practical preparation of trimethoprim: a classical antibacterial agent.syn. commun. 2013, 43, 1517–1522. jiang ja, du cy, gu ch, ji yf*. “one-pot” synthesis of 4-substituted 1,5-diaryl-1h-pyrazole-3- carboxylic acids via a meona/licl-mediated sterically hindered claisen condensation-knorr reaction-hydrolysis sequence. synlett 2012,23, 2965–2968. jiang ja, zhai jj, yu xh, teng x, ji yf*. a practical synthesis of cefcapene pivoxil. synthesis2012, 44, 207–214.
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